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Dergiler / Turkish Journal of Chemistry / 2017 / Cilt: 41 - Sayı: 3

Stereoselective and regioselective synthesis of NN-substituted methyl 2-((azolyl)methyl)-3-arylacrylates from Baylis-Hillman acetates

İlhami ÇELİK
Ayşen KÖSECELİ ÖZENÇ
Şule KÖKTEN
Sayfa
323–334
Yayın Tarihi
2022-11-05
DOI
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The targeted N -substituted azole acrylates were efficiently obtained in good yields (39% 89%).

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Amaç & Hipotez:N -Substituted methyl 2-((azolyl)methyl)-3-arylacrylates were synthesized stereo- and regioselectively with one-pot reaction between Baylis Hillman acetates and a suitable acylazole in the presence of K2 CO3 as a base catalyst.
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Temel Bulgular & Veri:N -Substituted methyl 2-((azolyl)methyl)-3-arylacrylates were synthesized stereo- and regioselectively with one-pot reaction between Baylis Hillman acetates and a suitable acylazole in the presence of K2 CO3 as a base catalyst.
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Sonuç & Katkı:The targeted N -substituted azole acrylates were efficiently obtained in good yields (39% 89%).
🔬Tür:Araştırma Makalesi
📍Kapsam:Genişletilmiş Akademik Örneklem
⚙️Değişkenler:Alan Parametreleri

Abstract

N -Substituted methyl 2-((azolyl)methyl)-3-arylacrylates were synthesized stereo- and regioselectively with one-pot reaction between Baylis Hillman acetates and a suitable acylazole in the presence of K2 CO3 as a base catalyst. The targeted N -substituted azole acrylates were efficiently obtained in good yields (39% 89%).

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Bu Makaleye Atıf Yap

ÇELİK, İ., ÖZENÇ, A. K., KÖKTEN, Ş. (2022). Stereoselective and regioselective synthesis of NN-substituted methyl 2-((azolyl)methyl)-3-arylacrylates from Baylis-Hillman acetates. Turkish Journal of Chemistry, Cilt: 41 - Sayı: 3, 323–334. https://ajindex.com/articles/601936

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