Dergiler / Turkish Journal of Chemistry / 2013 / Cilt: 37 - Sayı: 1

Synthesis, characterization, and antimicrobial activity of some new phosphorus macrocyclic compounds containing pyrazole rings

Sayfa
160–169
Yayın Tarihi
2013-01-01
DOI
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The antimicrobial activities of the synthesized compounds were assayed.

📌 3 Maddede Bu Makale

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Amaç & Hipotez:A simple synthetic method is reported for the preparation of some new phosphorus macrocycles in which the pyrazole rings are appended to a phosphorus atom.
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Temel Bulgular & Veri:The methodology is based on the cyclocondensation reaction of bis(4-formylpyrazolyl) phosphine oxide(1a, 1b) with nitrogen nucleophiles that contain active terminal amino groups.
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Sonuç & Katkı:The antimicrobial activities of the synthesized compounds were assayed.
🔬Tür:Araştırma Makalesi
📍Kapsam:Genişletilmiş Akademik Örneklem
⚙️Değişkenler:Key words: Phosphorus macrocycles · pyrazole · cyclocondensation

Özet

A simple synthetic method is reported for the preparation of some new phosphorus macrocycles in which the pyrazole rings are appended to a phosphorus atom. The methodology is based on the cyclocondensation reaction of bis(4-formylpyrazolyl) phosphine oxide(1a, 1b) with nitrogen nucleophiles that contain active terminal amino groups. The antimicrobial activities of the synthesized compounds were assayed.

Abstract

A simple synthetic method is reported for the preparation of some new phosphorus macrocycles in which the pyrazole rings are appended to a phosphorus atom. The methodology is based on the cyclocondensation reaction of bis(4-formylpyrazolyl) phosphine oxide(1a, 1b) with nitrogen nucleophiles that contain active terminal amino groups. The antimicrobial activities of the synthesized compounds were assayed.

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Bu Makaleye Atıf Yap

ALI, T. E., ABDEL-GHAFFAR, S. A., EL-MAHDY, K. M., ABDEL-KARIM, S. M. (2013). Synthesis, characterization, and antimicrobial activity of some new phosphorus macrocyclic compounds containing pyrazole rings. Turkish Journal of Chemistry, Cilt: 37 - Sayı: 1, 160–169. https://ajindex.com/articles/184813

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