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Dergiler / Turkish Journal of Chemistry / 2018 / Cilt: 42 - Sayı: 5

Tetrahydropyridine: a promising heterocycle for pharmacologically active molecules

Noor-ul-Amin MOHSIN
Matloob AHMAD
Sayfa
1191–1216
Yayın Tarihi
2018-10-11
DOI
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Yapay Zeka Hızlı Bakış & Çıkarımlar

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⚡ TL;DR(1 Cümlede Hızlı Çıkarım)

In this review, we summarize the recent literature dealing with the bioactive nature of this important heterocycle.

📌 3 Maddede Bu Makale

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Amaç & Hipotez:The tetrahydropyridine (THP) ring system has received considerable focus due to its excellent ability to act as a pharmacophore.
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Temel Bulgular & Veri:It is recognized as a major constituent in natural alkaloids.
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Sonuç & Katkı:In this review, we summarize the recent literature dealing with the bioactive nature of this important heterocycle.
🔬Tür:Literatür & Derleme Çalışması
📍Kapsam:Genişletilmiş Akademik Örneklem
⚙️Değişkenler:Functionalized tetrahydropyridine · condensed tetrahydropyridine · multicomponent reaction

Abstract

The tetrahydropyridine (THP) ring system has received considerable focus due to its excellent ability to act as a pharmacophore. It is recognized as a major constituent in natural alkaloids. THP derivatives have been reported for a diverse range of biological activities. Recent synthetic works contain syntheses of monosubstituted, disubstituted, trisubstituted, highly functionalized, and condensed structures. In this review, we summarize the recent literature dealing with the bioactive nature of this important heterocycle.

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Bu Makaleye Atıf Yap

MOHSIN, N., AHMAD, M. (2018). Tetrahydropyridine: a promising heterocycle for pharmacologically active molecules. Turkish Journal of Chemistry, Cilt: 42 - Sayı: 5, 1191–1216. https://ajindex.com/articles/184285

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