Journals / Turkish Journal of Chemistry / 2008 / Cilt: 32 - Sayı: 6

Synthesis and biological activity of allosteric modulators of $GABA_B$ receptors. Part 4. synthesis of potentially fluorescent acridines and conformationally restricted N-(arylpropyl)-1-arylethylamines

Pages
755–763
DOI
—

Abstract

A series of 8 new derivatives of fendiline was prepared for evaluation as allosteric modulators of $GABA_B$ receptors: 4 based on acridine and 4 with restricted distance between the 2 aryl moieties.