The results showed that some compounds had good insecticidal and bactericidal activity, e.g., the activities of compounds 6e and 6g–6j toward tobacco bacterial wilt were much better than those of commercial thiodiazole-copper, and some of the synthesized compounds possessed good insecticidal activity against Plutella xylostella.
📌 3 Key Takeaways
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Objective & Hypothesis:A series of novel sulfide derivatives containing 1,3,4-oxadiazole and pyridine were synthesized, characterized,and tested for their antibacterial activity against tobacco bacterial wilt and rice bacterial blight and for insecticidalactivity toward diamondback moth.
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Key Findings & Data:The results showed that some compounds had good insecticidal and bactericidal activity, e.g., the activities of compounds 6e and 6g–6j toward tobacco bacterial wilt were much better than those of commercial thiodiazole-copper, and some of the synthesized compounds possessed good insecticidal activity against Plutella xylostella.
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Conclusion & Impact:Compounds 6d, 6h, 6j, 6l, 6p, 6r, and 6p displayed over 93% activity at 500 mg L −1.
🔬Design:Research Article
📍Scope:Comprehensive Sample
⚙️Variables:Domain Parameters
Abstract
A series of novel sulfide derivatives containing 1,3,4-oxadiazole and pyridine were synthesized, characterized,and tested for their antibacterial activity against tobacco bacterial wilt and rice bacterial blight and for insecticidalactivity toward diamondback moth. The results showed that some compounds had good insecticidal and bactericidal activity, e.g., the activities of compounds 6e and 6g–6j toward tobacco bacterial wilt were much better than those of commercial thiodiazole-copper, and some of the synthesized compounds possessed good insecticidal activity against Plutella xylostella. Compounds 6d, 6h, 6j, 6l, 6p, 6r, and 6p displayed over 93% activity at 500 mg L −1.
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Cite This Article
CHEN, S., HE, F., ZHANG, Y., LUO, D., WU, J., YU, G. (2022). Synthesis and bioactivity of sulfide derivatives containing 1,3,4-oxadiazole and pyridine. Turkish Journal of Chemistry, Cilt: 43 - Sayı: 4, 1075–1085. https://ajindex.com/articles/601714
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